Synthetic chemistry plays a central role in many areas of chemical biology; utilising recent case studies, the goal of is to highlight the full impact that the preparation of novel reagents can have in chemical biology. Covering the synthetic approaches that can be applied across the whole field of chemical biology, this book provides synthetic chemists with the broader context to which their work contributes and the biological questions that can be addressed through it. An ideal guide for postgraduate students and researchers in synthetic organic chemistry and chemical biology, introduces synthetic techniques and methods to those who wish to incorporate synthesis for the first time in their biology-focused research programmes.